Search on: STAUROSPORINE 
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Descriptor English:   Staurosporine 
Descriptor Spanish:   Estaurosporina 
Descriptor Portuguese:   Estaurosporina 
Tree Number:   D03.132.436.750
D03.633.100.473.144.750
D03.633.100.473.402.750
D03.633.300.148.750
Definition English:   An indolocarbazole that is a potent PROTEIN KINASE C inhibitor which enhances cAMP-mediated responses in human neuroblastoma cells. (Biochem Biophys Res Commun 1995;214(3):1114-20) 
Pharmacological Action:   Enzyme Inhibitors
 
History Note English:   97; was STAUROSPORINE (NM) 1977-96 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AA analogs & derivatives
AN analysis AI antagonists & inhibitors
BI biosynthesis BL blood
CF cerebrospinal fluid CS chemical synthesis
CH chemistry CL classification
CT contraindications DF deficiency
EC economics GE genetics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PH physiology PO poisoning
RE radiation effects SE secretion
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UR urine  
Record Number:   32990 
Unique Identifier:   D019311 

Occurrence in VHL:
 

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